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Drug Classifications
Drug Classifications
5-alpha reductase inhibitor
1 Subclass
Type I and Type II isoenzyme inhibitor
1 Drug
5α-reductase inhibitor
1 Subclass
Type II 5α-reductase inhibitor
1 Drug
Acid Suppressant
1 Subclass
Potassium-Competitive Acid Blocker (P-CAB)
1 Drug
Adrenal enzyme inhibitor
1 Subclass
Steroidogenesis inhibitor
1 Drug
Alcohol Dependence Treatment Agent
1 Subclass
GABA/Glutamate Modulator
1 Drug
Alcohol Deterrent
1 Subclass
Aldehyde Dehydrogenase Inhibitor
1 Drug
Aldosterone antagonist
1 Subclass
Potassium-sparing diuretic (active metabolite of spironolactone)
1 Drug
Alkalinising Agent
1 Subclass
Systemic Electrolyte Modifier
1 Drug
Alkylating agent
1 Subclass
Nitrogen mustard derivative
1 Drug
Alpha-adrenergic antagonist
1 Subclass
Selective alpha-1A adrenergic receptor blocker
1 Drug
Analgesic
1 Subclass
Centrally-acting Weak Opioid Analgesic (Atypical Opioid)
1 Drug
Analgesic and Antipyretic
1 Subclass
Non-opioid Analgesic (Para-aminophenol Derivative)
1 Drug
Antacid
1 Subclass
Aluminium-containing non-systemic antacid
1 Drug
Antacid / Laxative
1 Subclass
Inorganic Magnesium Salt (Saline Laxative / Neutralizing Antacid)
1 Drug
Anthelmintic
2 Subclasses
Anti-filarial agent
1 Drug
Antischistosomal / Anticestodal
1 Drug
Anti-anginal Agent
2 Subclasses
Long-acting Nitrate Vasodilator
1 Drug
Potassium Channel Activator with Nitrate-like Properties
1 Drug
Anti-asthmatic / Anti-allergic
1 Subclass
Leukotriene Receptor Antagonist (LTRA)
1 Drug
Anti-inflammatory (Gastrointestinal)
1 Subclass
5-Aminosalicylic Acid (5-ASA) derivative
2 Drugs
Anti-inflammatory (GI)
1 Subclass
5-Aminosalicylic Acid (5-ASA) Prodrug
1 Drug
Anti-inflammatory (Non-steroidal)
1 Subclass
Selective Phosphodiesterase-4 (PDE-4) Inhibitor
1 Drug
Anti-inflammatory / Immunomodulatory
1 Subclass
5-Aminosalicylate derivative
1 Drug
Anti-inflammatory agent
1 Subclass
Microtubule polymerization inhibitor
1 Drug
Anti-inflammatory Agents
1 Subclass
5-Aminosalicylic Acid (5-ASA) Derivatives
1 Drug
Anti-inflammatory Dermatologic Agent
1 Subclass
Non-steroidal Phosphodiesterase-4 (PDE4) Inhibitor
1 Drug
Anti-resorptive agent
1 Subclass
RANKL (Receptor Activator of Nuclear Factor Kappa-B Ligand) Inhibitor
1 Drug
Antiacne agent
1 Subclass
Dicarboxylic acid derivative
1 Drug
Antiallergic / Anti-inflammatory
1 Subclass
H1-antihistamine (non-selective); Mast cell stabiliser
1 Drug
Antiallergic Agent
1 Subclass
Mast Cell Stabiliser
2 Drugs
Antiallergic agents
1 Subclass
Leukotriene receptor antagonist + Second-generation antihistamine
1 Drug
Antianginal
1 Subclass
Nitrate Vasodilator
1 Drug
Antianginal Agent
2 Subclasses
Metabolic Modulator (Fatty Acid Oxidation Inhibitor)
1 Drug
Metabolic Modulator (Late Sodium Current Inhibitor)
1 Drug
Antiarrhythmic
3 Subclasses
Class IB Sodium Channel Blocker
1 Drug
Class III antiarrhythmic (also non-selective beta-blocker)
1 Drug
Class III Antiarrhythmic (Potassium Channel Blocker)
1 Drug
Antiarrhythmic agent
1 Subclass
Nucleoside/purine receptor agonist (Class V antiarrhythmic)
1 Drug
Antibacterial
30 Subclasses
2nd Generation Oral Cephalosporin
1 Drug
3rd Generation Oral Cephalosporin
2 Drugs
Aminoglycoside
2 Drugs
Amphenicol antibiotic
1 Drug
Beta-lactam — Penem (Oral Penem)
1 Drug
Beta-lactam — Penicillinase-resistant Penicillin
3 Drugs
Carbapenem (Imipenem) + Renal Dehydropeptidase-I Inhibitor (Cilastatin)
1 Drug
Carbapenem (β-lactam)
1 Drug
Cyclic Lipopeptide Antibiotic
1 Drug
Extended-spectrum penicillin (Ureidopenicillin)
1 Drug
Extended-spectrum penicillin + Beta-lactamase inhibitor combination
1 Drug
First-generation Cephalosporin
3 Drugs
Fluoroquinolone (4th generation)
1 Drug
Fourth-generation cephalosporin
1 Drug
Fourth-Generation Cephalosporin (Anti-pseudomonal)
No Drugs
Glycylcycline (Tetracycline Derivative)
1 Drug
Lincosamide
1 Drug
Lipoglycopeptide antibiotic
1 Drug
Macrocyclic Antibiotic
1 Drug
Macrolide antibiotic
3 Drugs
Monobactam Beta-Lactam Antibiotic
1 Drug
Oxazolidinone
2 Drugs
Penicillin + Beta-lactamase inhibitor combination
1 Drug
Polymyxins (Cationic polypeptide antibiotics)
1 Drug
Tetracycline antibiotic
1 Drug
Third-Generation Cephalosporin
3 Drugs
Third-Generation Cephalosporin (Anti-pseudomonal)
1 Drug
Third-generation oral cephalosporin
1 Drug
Topical Antibiotic (Pseudomonic Acid Derivative)
1 Drug
Urinary antiseptic (Nitrofuran derivative)
1 Drug
Antibacterial + Antiprotozoal combination
2 Subclasses
Beta-lactam antibiotic + Nitroimidazole derivative
1 Drug
Penicillin (β-lactam) + Nitroimidazole
1 Drug
Antibacterial Agent
0 Drugs
Antibacterial combination
1 Subclass
Nitroimidazole derivative + Fluoroquinolone
1 Drug
Antibacterials
2 Subclasses
Non-systemic rifamycin derivative
1 Drug
Third-generation cephalosporin + Fluoroquinolone combination
2 Drugs
Antibiotic
12 Subclasses
Aminoglycoside antibiotic
4 Drugs
Fifth-generation Cephalosporin
1 Drug
Fluoroquinolone (Respiratory Fluoroquinolone)
1 Drug
Glycopeptide antibiotic
2 Drugs
Lipoglycopeptide
1 Drug
Phosphonic acid derivative
1 Drug
Pleuromutilin
1 Drug
Polymyxin (Polymyxin E)
1 Drug
Siderophore Cephalosporin
1 Drug
Sulfonamide + Dihydrofolate Reductase Inhibitor (Fixed-Dose Combination)
1 Drug
Tetracycline group
1 Drug
Third-generation cephalosporin (oral)
1 Drug
Antibiotic
1 Subclass
Second-generation cephalosporin
1 Drug
Anticholinergic
2 Subclasses
Antimuscarinic agent (quaternary ammonium compound)
1 Drug
Mydriatic and Cycloplegic Agent
1 Drug
Anticholinergic (Parasympatholytic)
1 Subclass
Muscarinic receptor antagonist
1 Drug
Anticoagulant
6 Subclasses
Direct Oral Anticoagulant (DOAC) — Factor Xa inhibitor
3 Drugs
Direct Thrombin Inhibitor
1 Drug
Indirect thrombin inhibitor (via antithrombin III potentiation)
1 Drug
Low Molecular Weight Heparin (Factor Xa inhibitor predominant)
1 Drug
Selective Factor Xa Inhibitor (Synthetic Pentasaccharide)
1 Drug
Vitamin K Antagonist (Coumarin derivative)
1 Drug
Anticonvulsant
3 Subclasses
GABA Analogue (Gabapentinoid)
1 Drug
Iminostilbene derivative
1 Drug
Phenyltriazine Derivative
1 Drug
Anticonvulsant / Anxiolytic
1 Subclass
Benzodiazepine (long-acting)
2 Drugs
Anticonvulsant / Neuropathic Pain Agent
1 Subclass
Alpha-2-delta Calcium Channel Ligand
1 Drug
Antidepressant
13 Subclasses
Melatonergic Agonist with 5-HT2C Antagonist Activity
1 Drug
Noradrenergic and Specific Serotonergic Antidepressant (NaSSA)
1 Drug
Norepinephrine-Dopamine Reuptake Inhibitor (NDRI)
1 Drug
Reversible Inhibitor of Monoamine Oxidase A (RIMA)
1 Drug
Selective Noradrenaline Reuptake Inhibitor (NaRI)
1 Drug
Selective Serotonin Reuptake Inhibitor (SSRI)
5 Drugs
Serotonin Antagonist and Reuptake Inhibitor (SARI)
1 Drug
Serotonin Modulator and Stimulator (SMS)
1 Drug
Serotonin-Norepinephrine Reuptake Inhibitor (SNRI)
3 Drugs
SSRI and 5-HT1A receptor partial agonist
1 Drug
Tetracyclic Antidepressant (TeCA)
1 Drug
Tricyclic Antidepressant (TCA)
7 Drugs
Tricyclic Antidepressant (TCA) — Dibenzoxazepine Group
1 Drug
Antidiabetic
12 Subclasses
Dipeptidyl Peptidase-4 (DPP-4) Inhibitor
6 Drugs
DPP-4 (Dipeptidyl Peptidase-4) Inhibitor
1 Drug
GLP-1 Receptor Agonist
1 Drug
GLP-1 Receptor Agonist (Incretin Mimetic)
3 Drugs
Long-acting Insulin Analogue
1 Drug
Rapid-acting insulin analogue
2 Drugs
SGLT2 inhibitor (Sodium-glucose co-transporter 2 inhibitor
1 Drug
Short-acting human insulin
1 Drug
Sodium-Glucose Co-Transporter-2 (SGLT2) Inhibitor
1 Drug
Sulfonylurea (first-generation)
3 Drugs
Sulfonylurea (second-generation)
4 Drugs
Thiazolidinedione (Insulin Sensitizer)
1 Drug
Antidiabetic / Antilipidemic
1 Subclass
Dual PPAR α/γ Agonist (Glitazar class)
1 Drug
Antidiabetic Agent
8 Subclasses
Alpha-Glucosidase Inhibitor
3 Drugs
Biguanide
1 Drug
Biphasic insulin (Intermediate-acting + Short-acting human insulin)
1 Drug
Glucagon-Like Peptide-1 (GLP-1) Receptor Agonist
1 Drug
Long-acting basal insulin analogue
1 Drug
Meglitinide (Short-Acting Insulin Secretagogue)
1 Drug
Sodium-Glucose Cotransporter 2 (SGLT2) Inhibitor
2 Drugs
Thiazolidinedione (PPAR-γ Agonist)
1 Drug
Antidiarrhoeal
2 Subclasses
Enkephalinase inhibitor
1 Drug
Peripheral opioid receptor agonist
1 Drug
Antidote
1 Subclass
Immunoglobulin fragment (Fab) – Digitalis Antidote
1 Drug
Antidote / Mucolytic
1 Subclass
Glutathione Precursor (Sulfhydryl Donor)
1 Drug
Antidyskinetic Agent
1 Subclass
Vesicular Monoamine Transporter 2 (VMAT2) Inhibitor
1 Drug
Antiemetic
6 Subclasses
5-HT3 (Serotonin) receptor antagonist
1 Drug
5-HT₃ (Serotonin) Receptor Antagonist
1 Drug
5-HT3 receptor antagonist
1 Drug
Antihistamine (H1 receptor antagonist)
1 Drug
Neurokinin-1 (NK1) Receptor Antagonist
1 Drug
Phenothiazine Dopamine Antagonist
1 Drug
Antiepileptic
17 Subclasses
AMPA Receptor Antagonist (Selective Non-competitive Antagonist at α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid Receptor)
1 Drug
Barbiturate
1 Drug
Barbiturate-related anticonvulsant
1 Drug
Benzodiazepine (1,5-benzodiazepine)
1 Drug
Broad-spectrum anticonvulsant (valproate group)
1 Drug
Dibenzazepine Carboxamide Derivative
1 Drug
Functionalized Amino Acid (Sodium Channel Modulator)
1 Drug
GABA-transaminase inhibitor
1 Drug
GABAergic, Enzyme Inhibitor
1 Drug
Hydantoin derivative
1 Drug
Pyrrolidone derivative
1 Drug
Sodium channel blocker (dibenzoazepine derivative)
1 Drug
Succinimide derivative
1 Drug
Sulfamate-substituted Monosaccharide Derivative
1 Drug
Sulfonamide-Based Anticonvulsant
1 Drug
SV2A (Synaptic Vesicle Protein 2A) Ligand
1 Drug
Triazole Derivative Anticonvulsant
1 Drug
Antiepileptic (AED)
2 Subclasses
Dicarbamate anticonvulsant
1 Drug
GABA Reuptake Inhibitor
1 Drug
Antifibrinolytic
1 Subclass
Synthetic lysine analogue
1 Drug
Antifibrotic agent
1 Subclass
Pyridone derivative
1 Drug
Antifungal
7 Subclasses
Antifungal – Systemic (for dermatophytosis)
1 Drug
Echinocandin
2 Drugs
Imidazole derivative
1 Drug
Imidazole Derivative (Azole Antifungal)
1 Drug
Morpholine derivative antifungal
1 Drug
Pyrimidine Analogue
1 Drug
Triazole antifungal
3 Drugs
Antifungal agent
1 Subclass
Polyene antifungal
2 Drugs
Antiglaucoma agent
2 Subclasses
Alpha-2 adrenergic receptor agonist
1 Drug
Carbonic Anhydrase Inhibitor (Topical)
1 Drug
Antigout agent
0 Drugs
Antihistamine
9 Subclasses
First-generation H1 receptor antagonist
2 Drugs
First-generation H1 receptor antagonist (with anxiolytic and sedative properties)
1 Drug
First-generation H1 receptor antagonist; Anticholinergic
1 Drug
Second-Generation H1 Antihistamine (Non-sedating/Low-sedating)
1 Drug
Second-Generation H1 Receptor Antagonist
1 Drug
Second-generation H1-receptor antagonist (minimally sedating antihistamine)
1 Drug
Second-generation H1-receptor antagonist (piperazine derivative)
No Drugs
Second-generation non-sedating H1-receptor antagonist
2 Drugs
Selective H1-receptor antagonist (second-generation, non-sedating antihistamine)
1 Drug
Antihistamine (First-generation)
1 Subclass
Phenothiazine derivative
1 Drug
Antihistamine / Antiallergic Agent
1 Subclass
Selective H1 Receptor Antagonist with Mast Cell Stabilising Activity
1 Drug
Antihyperlipidaemic
2 Subclasses
Bile Acid Sequestrant
1 Drug
Nicotinic acid derivative
1 Drug
Antihypertensive
16 Subclasses
Alpha-1 adrenergic receptor antagonist
1 Drug
Alpha-1 adrenergic receptor blocker
1 Drug
Angiotensin-Converting Enzyme (ACE) Inhibitor
5 Drugs
Calcium Channel Blocker — Dihydropyridine (L-type and N-type)
1 Drug
Calcium Channel Blocker — Dihydropyridine class
1 Drug
Centrally acting alpha-2 adrenergic agonist
2 Drugs
Combined alpha- and beta-adrenergic receptor blocker
1 Drug
Dihydropyridine Calcium Channel Blocker (2nd generation)
1 Drug
Dihydropyridine Calcium Channel Blocker (DHP-CCB)
1 Drug
Dihydropyridine Calcium Channel Blocker (third-generation)
1 Drug
Direct Renin Inhibitor
1 Drug
Direct-acting arteriolar vasodilator
1 Drug
Non-selective Beta-blocker with Intrinsic Sympathomimetic Activity (ISA)
1 Drug
Non-selective, Irreversible Alpha-Adrenergic Blocker
1 Drug
Sympatholytic (Adrenergic Neuron Blocker)
1 Drug
Thiazide-like diuretic
2 Drugs
Antihypertensive (oral) / Hair Growth Promoter (topical)
1 Subclass
Potassium Channel Opener / Vasodilator
1 Drug
Antihypertensive / Antianginal Agent
1 Subclass
Dihydropyridine Calcium Channel Blocker (CCB)
1 Drug
Antihypertensive / Nephroprotective Agent
1 Subclass
Angiotensin II Receptor Blocker (ARB)
5 Drugs
Antihypertensive agent
1 Subclass
Centrally acting imidazoline receptor agonist (I₁-receptor agonist)
1 Drug
Antilipidemic
1 Subclass
Fibrate (Fibric Acid Derivative)
2 Drugs
Antimalarial / Disease-Modifying Antirheumatic Drug (DMARD)
1 Subclass
4-Aminoquinoline derivative
1 Drug
Antimetabolite
1 Subclass
Folate Antagonist / Disease-Modifying Antirheumatic Drug (DMARD)
1 Drug
Antimicrobial
6 Subclasses
Antitubercular Agent (First-line)
1 Drug
Fluoroquinolone
2 Drugs
Nitroimidazole anti-protozoal and anaerobic antibacterial
1 Drug
Nitroimidazole derivative
1 Drug
Nitroimidazole derivative (antiprotozoal and anaerobic antibacterial)
2 Drugs
Sulfone antibiotic
1 Drug
Antimicrobial + Probiotic
1 Subclass
Tetracycline-class antibiotic + Live microbial supplement
1 Drug
Antimigraine
1 Subclass
5-HT1B/1D Receptor Agonist (Triptan)
1 Drug
Antimigraine agent
2 Subclasses
Selective 5-HT1B/1D receptor agonist (Triptan)
1 Drug
Serotonin (5-HT1B/1D) receptor agonist (Triptan)
1 Drug
Antimitotic Agent
1 Subclass
Topical Cytotoxic (Plant-derived)
1 Drug
Antimuscarinic
0 Drugs
Antimuscarinic (Anticholinergic)
1 Subclass
M3-Selective Muscarinic Receptor Antagonist
1 Drug
Antimuscarinic agent
1 Subclass
Urinary antispasmodic
2 Drugs
Antimycobacterial
8 Subclasses
Anti-tubercular agent (Nitroimidazo-oxazole derivative)
1 Drug
Diarylquinoline antimycobacterial
1 Drug
First-line Antitubercular Agent
1 Drug
Rifamycin antibiotic
1 Drug
Second-line Anti-TB Drug (Group C – WHO classification)
1 Drug
Second-line Anti-TB Drug (Group C – WHO/ICMR classification)
1 Drug
Second-line Antitubercular Agent
2 Drugs
Thioamide (Second-line Antitubercular Agent)
1 Drug
Antimycobacterial agent
1 Subclass
Rifamycin derivative
2 Drugs
Antineoplastic
2 Subclasses
Tyrosine Kinase Inhibitor (BCR-ABL, c-KIT, PDGFR)
1 Drug
Tyrosine kinase inhibitor (TKI) — multi-targeted (VEGFR, MET, AXL, RET)
1 Drug
Antineoplastic / Haemoglobin modulator
1 Subclass
Antimetabolite (ribonucleotide reductase inhibitor)
1 Drug
Antineoplastic agent
7 Subclasses
Adrenal Cytotoxic Agent
1 Drug
Anthracycline Antibiotic
1 Drug
Aromatase inhibitor (non-steroidal)
1 Drug
Cytotoxic Antibiotic (Antitumour Antibiotic)
1 Drug
Platinum-based Alkylating Agent
1 Drug
Platinum-based Alkylating-like Compound
1 Drug
Topoisomerase II Inhibitor
1 Drug
Antiparasitic
2 Subclasses
Antiprotozoal / Broad-spectrum Antiparasitic
1 Drug
Avermectin macrocyclic lactone
1 Drug
Antiparkinsonian
6 Subclasses
Catechol-O-Methyltransferase (COMT) Inhibitor
2 Drugs
Dopa Decarboxylase Inhibitor (DDCI)
1 Drug
Dopamine Agonist (Non-ergot derived; D2/D3 receptor agonist)
1 Drug
Dopamine Agonist (Non-ergot derived)
1 Drug
Dopaminergic agent (dopamine precursor)
1 Drug
Selective MAO-B Inhibitor
1 Drug
Antiparkinsonian Agent
3 Subclasses
Anticholinergic (Muscarinic Antagonist)
1 Drug
Centrally Acting Anticholinergic (Muscarinic Antagonist)
1 Drug
Monoamine Oxidase-B (MAO-B) Inhibitor
1 Drug
Antiplatelet
1 Subclass
P2Y12 ADP Receptor Inhibitor
1 Drug
Antiplatelet / Vasodilator
1 Subclass
Phosphodiesterase Inhibitor (Non-selective)
1 Drug
Antiplatelet agent
4 Subclasses
Glycoprotein IIb/IIIa receptor antagonist
2 Drugs
Glycoprotein IIb/IIIa Receptor Inhibitor
1 Drug
P2Y12 ADP receptor inhibitor (Thienopyridine)
1 Drug
P2Y12 Receptor Antagonist (Reversible, Direct-acting)
1 Drug
Antiplatelet agent / Analgesic / Antipyretic
1 Subclass
Non-steroidal anti-inflammatory drug (NSAID), Salicylate
1 Drug
Antipsychotic
14 Subclasses
Atypical (Second-Generation) Antipsychotic
4 Drugs
Atypical (second-generation) antipsychotic – Dopamine D3/D2 partial agonist
1 Drug
Atypical (Second-generation) Antipsychotic – Thienobenzodiazepine derivative
1 Drug
Atypical (Second-Generation) Antipsychotic — Dopamine Partial Agonist
1 Drug
Atypical (Substituted Benzamide)
1 Drug
Diphenylbutylpiperidine (Typical/First-generation Antipsychotic)
1 Drug
First-generation (typical) antipsychotic – Butyrophenone derivative
1 Drug
First-Generation (Typical) Antipsychotic — Phenothiazine (Aliphatic subgroup)
1 Drug
First-Generation (Typical) Antipsychotic — Phenothiazine (Piperazine subgroup)
1 Drug
Second-generation (atypical) antipsychotic
1 Drug
Substituted Benzamide (Selective Dopamine D2/D3 Antagonist)
1 Drug
Typical (First-generation) Antipsychotic – Phenothiazine group
1 Drug
Typical (First-generation) Antipsychotic — Thioxanthene Derivative
1 Drug
Typical (First-Generation) Antipsychotic — Thioxanthene Group
1 Drug
Antiretroviral
3 Subclasses
Integrase Strand Transfer Inhibitor (INSTI)
1 Drug
Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI)
2 Drugs
Protease Inhibitor (PI)
1 Drug
Antispasmodic
3 Subclasses
Anticholinergic (Antimuscarinic)
1 Drug
Muscarinic Antagonist (Peripherally Acting Anticholinergic)
1 Drug
Selective phosphodiesterase-4 inhibitor (non-cholinergic, non-opioid antispasmodic)
1 Drug
Antithyroid agent
2 Subclasses
Thioamide derivative
1 Drug
Thionamide derivative
1 Drug
Antitubercular agent
2 Subclasses
First-line antimycobacterial (bactericidal)
1 Drug
Nitroimidazooxazine derivative
1 Drug
Antiulcer agent
0 Drugs
Antivertigo / Antihistamine
1 Subclass
Piperazine derivative
1 Drug
Antivertigo Agent / Histamine Analogue
1 Subclass
H1 Receptor Agonist and H3 Receptor Antagonist
1 Drug
Antiviral
11 Subclasses
Anti-CMV Agent (Nucleoside Analogue Prodrug)
1 Drug
Anti-CMV Agent (Nucleoside Analogue)
1 Drug
Direct-Acting Antiviral (DAA) – NS5B Polymerase Inhibitor
1 Drug
HIV Integrase Strand Transfer Inhibitor (INSTI)
1 Drug
Neuraminidase Inhibitor
1 Drug
Nucleoside Analogue (Anti-HBV)
1 Drug
Nucleoside analogue (Guanine derivative)
1 Drug
Nucleoside Reverse Transcriptase Inhibitor (NRTI)
2 Drugs
Nucleotide Reverse Transcriptase Inhibitor (NtRTI)
1 Drug
Protease Inhibitor (PI) — Antiretroviral
1 Drug
Protease Inhibitor (PI) — Antiretroviral
1 Drug
Antiviral agents
0 Drugs
Antiviral and Antiparkinsonian agent
1 Subclass
Adamantane derivative (dopaminergic agonist and NMDA receptor antagonist)
1 Drug
Anxiolytic
2 Subclasses
Azapirone Derivative (5-HT1A Partial Agonist)
1 Drug
Benzodiazepine — Short-acting
1 Drug
Anxiolytic / Sedative-Hypnotic
1 Subclass
Benzodiazepine (intermediate-acting)
1 Drug
Atypical Antipsychotic
4 Subclasses
Benzisothiazole Derivative
2 Drugs
Dibenzothiazepine derivative
1 Drug
Serotonin-dopamine activity modulator
1 Drug
Serotonin-Dopamine Antagonist (SDA)
1 Drug
Benzodiazepine
2 Subclasses
Hypnotic Benzodiazepine (Long-acting)
1 Drug
Short-acting hypnotic/anxiolytic
1 Drug
Beta-adrenergic blocker
2 Subclasses
Cardioselective beta-1 blocker (ultra-short acting)
1 Drug
Non-selective beta-blocker
2 Drugs
Beta-adrenergic blocker (Beta-blocker)
2 Subclasses
Beta-1 selective adrenergic receptor blocker with nitric oxide-mediated vasodilatory property
1 Drug
Cardioselective beta-1 blocker
1 Drug
Beta-adrenoceptor Antagonist
1 Subclass
Cardioselective β1-blocker with Intrinsic Sympathomimetic Activity (ISA)
1 Drug
Beta-adrenoceptor blocker
1 Subclass
Cardioselective β1-blocker
1 Drug
Beta-adrenoceptor Blocker (Beta-blocker)
1 Subclass
Beta-1 Selective (Cardioselective) Beta-blocker
1 Drug
Beta-blocker
1 Subclass
Non-selective beta-adrenergic antagonist
1 Drug
Beta-lactamase inhibitor
1 Subclass
Penicillanic acid sulfone beta-lactamase inhibitor
1 Drug
Bone Metabolism Regulator
2 Subclasses
Bisphosphonate (Nitrogen-Containing)
2 Drugs
Hormonal Agent / Calcitonin Analogue
1 Drug
Bone-forming agent
1 Subclass
Recombinant human parathyroid hormone analog (PTH 1–34)
1 Drug
Bronchodilator
12 Subclasses
Anticholinergic (Short-Acting Muscarinic Antagonist — SAMA)
1 Drug
Long-acting beta-2 adrenergic agonist (LABA)
1 Drug
Long-acting beta-2 adrenergic agonist (LABA) – prodrug of terbutaline
1 Drug
Long-Acting Beta-2 Agonist (LABA)
1 Drug
Long-acting muscarinic antagonist (LAMA)
1 Drug
Long-acting β2-adrenergic receptor agonist (LABA)
1 Drug
Long-acting β2-agonist (LABA)
1 Drug
Methylxanthine derivative
1 Drug
Non-selective phosphodiesterase inhibitor (PDE3 and PDE4), anti-inflammatory
1 Drug
Selective β2-adrenergic receptor agonist
1 Drug
Short-acting β2-adrenergic receptor agonist (SABA)
1 Drug
Xanthine derivative + Mucoregulator (Ambroxol derivative)
1 Drug
Calcium Channel Blocker
3 Subclasses
Dihydropyridine
2 Drugs
Non-dihydropyridine (benzothiazepine-type)
1 Drug
Phenylalkylamine (non-dihydropyridine)
1 Drug
Calcium Channel Blocker (Antihypertensive)
1 Subclass
Dihydropyridine Calcium Channel Blocker
1 Drug
Calcium channel blocker (non-selective)
1 Subclass
Cerebral vasodilator / Antimigraine / Vestibular suppressant
1 Drug
Calcium Homeostasis Regulator
1 Subclass
Calcimimetic Agent
1 Drug
Carbonic Anhydrase Inhibitor
1 Subclass
Diuretic / Antiglaucoma Agent / Antiepileptic
1 Drug
Cardiac Agent
1 Subclass
If Channel Inhibitor (Selective Sinus Node Inhibitor)
1 Drug
Cardiac glycoside
2 Subclasses
Digitalis alkaloid
1 Drug
Digitalis derivative
1 Drug
Cardiovascular Agent
3 Subclasses
Angiotensin receptor neprilysin inhibitor (ARNI)
1 Drug
Inodilator (Calcium sensitizer with potassium channel opening activity)
1 Drug
Selective Aldosterone Receptor Antagonist (Mineralocorticoid Receptor Antagonist — MRA)
1 Drug
Central Nervous System Stimulant
1 Subclass
Wakefulness-Promoting Agent
1 Drug
Cholinergic (Parasympathomimetic) Agent
5 Subclasses
Cholinesterase Inhibitor (Long-acting, Reversible)
1 Drug
Cholinesterase Inhibitor (Reversible)
2 Drugs
Cholinesterase Inhibitor (Short-acting, Reversible)
1 Drug
Muscarinic and Nicotinic Receptor Agonist
1 Drug
Muscarinic Receptor Agonist
3 Drugs
Cholinergic Agent
1 Subclass
Muscarinic Agonist (Direct-acting Parasympathomimetic)
No Drugs
Cholinesterase Inhibitor
1 Subclass
Reversible Anticholinesterase
1 Drug
CNS Agent
1 Subclass
NMDA Receptor Antagonist
1 Drug
Cognitive Enhancer
2 Subclasses
Acetylcholinesterase Inhibitor
1 Drug
Cholinesterase Inhibitor (Dual Acetylcholinesterase and Butyrylcholinesterase Inhibitor)
1 Drug
Corticosteroid
6 Subclasses
Glucocorticoid
2 Drugs
Glucocorticoid (Inhaled, Intranasal, Topical)
1 Drug
Glucocorticoid (Long-acting, High Potency)
1 Drug
Glucocorticoid (Synthetic, Non-halogenated)
1 Drug
Glucocorticoid (with significant mineralocorticoid activity)
1 Drug
Topical Corticosteroid — Super-Potent / Very High Potency (Group I / Class I)
1 Drug
Corticosteroid (Inhaled)
1 Subclass
Inhaled Glucocorticoid
2 Drugs
Dermatological Agent
5 Subclasses
Antipsoriatic (cytotoxic/antiproliferative)
1 Drug
Antipsoriatic / Keratoplastic
1 Drug
Skin protectant / Antipruritic
1 Drug
Topical Antimicrobial / Keratolytic Agent
1 Drug
Topical retinoid
1 Drug
Digestive enzymes
2 Subclasses
Pancreatic enzyme replacement
1 Drug
Pancreatic Enzyme Replacement Therapy (PERT)
1 Drug
Disease-Modifying Antirheumatic Drug (DMARD)
2 Subclasses
Janus Kinase (JAK) Inhibitor
2 Drugs
Pyrimidine synthesis inhibitor
1 Drug
Diuretic
3 Subclasses
Loop diuretic
3 Drugs
Potassium-sparing diuretic; Aldosterone antagonist
1 Drug
Thiazide Diuretic
1 Drug
Diuretic (Potassium-sparing)
1 Subclass
Epithelial Sodium Channel (ENaC) Inhibitor
1 Drug
Diuretic and Antihypertensive
1 Subclass
Thiazide-like Diuretic (Indoline derivative)
1 Drug
Dopamine agonist
1 Subclass
Ergot derivative
1 Drug
Dopaminergic agent
1 Subclass
Ergot-derived dopamine D2 receptor agonist
1 Drug
Ectoparasiticide
1 Subclass
Synthetic Pyrethroid Insecticide
1 Drug
Electrolyte and Fluid Replacement
1 Subclass
Oral Rehydration Salts (WHO reduced osmolarity formula)
1 Drug
Electrolyte replacement / Anticonvulsant
1 Subclass
Magnesium salt
1 Drug
Electrolyte supplement
1 Subclass
Potassium salt
1 Drug
Endocrine Therapy
1 Subclass
Growth Hormone Receptor Antagonist
1 Drug
Endothelin Receptor Antagonist
2 Subclasses
Dual (ETA and ETB) Endothelin Receptor Antagonist
1 Drug
Selective Endothelin-A (ETA) Receptor Antagonist
1 Drug
Gastrointestinal agent
5 Subclasses
Chloride channel activator (type-2 chloride channel agonist)
1 Drug
Cytoprotective / Mucosal protective agent
1 Drug
Guanylate cyclase-C agonist
1 Drug
Mixed Opioid Receptor Modulator
1 Drug
Mucosal protectant (Cytoprotective agent)
1 Drug
Gastrointestinal Protectants
1 Subclass
Mucosal Defense Enhancers
1 Drug
Gastroprokinetic agent
2 Subclasses
Dopamine D2 receptor antagonist with acetylcholinesterase inhibitory activity
1 Drug
Selective 5-HT4 Receptor Agonist
1 Drug
General anaesthetic
1 Subclass
Intravenous anaesthetic agent
1 Drug
Glucagon-like peptide-2 (GLP-2) analogue
1 Subclass
Intestinal growth factor
1 Drug
Glucocorticoid (local/rectal)
1 Subclass
Gastroenterology
1 Drug
Gonadotropin-Releasing Hormone (GnRH) Analog
1 Subclass
GnRH Agonist
1 Drug
H2-Receptor Antagonist
1 Drug
Gastric acid secretion inhibitor
1 Drug
Histamine H2 Blocker
1 Drug
Histamine-2 Receptor Blocker
1 Drug
Famotidine
Haematinic
2 Subclasses
Oral Iron Supplement
1 Drug
Oral Iron Supplement (Chelated Iron with Ascorbic Acid)
1 Drug
Haematopoietic agent
1 Subclass
Erythropoiesis-Stimulating Agent (ESA)
2 Drugs
Haematopoietic growth factor
1 Subclass
Granulocyte colony-stimulating factor (G-CSF)
1 Drug
Hemorheologic agent
1 Subclass
Xanthine derivative
1 Drug
Hepatobiliary agent
1 Subclass
Bile acid derivative
1 Drug
Hepatobiliary agents
1 Subclass
Farnesoid X receptor (FXR) agonist
1 Drug
Hormones
1 Subclass
Recombinant Human Growth Hormone (r-hGH)
1 Drug
Hormones and Antidotes
1 Subclass
Hyperglycaemic Agent
1 Drug
Hyperglycaemic / Antihypertensive
1 Subclass
Potassium channel activator (ATP-sensitive K⁺ channel opener)
1 Drug
Hypnotic
2 Subclasses
Cyclopyrrolone derivative (Z-drug)
1 Drug
Endogenous Hormone / Circadian Rhythm Regulator
1 Drug
Hypnotic/Sedative
1 Subclass
Non-benzodiazepine GABA-A Receptor Agonist (Z-drug)
1 Drug
Immunomodulator
8 Subclasses
Anti-IL-17A monoclonal antibody
1 Drug
Calcineurin inhibitor (Topical)
1 Drug
Interferons (Type I beta interferons)
1 Drug
Janus Kinase (JAK) 1 Selective Inhibitor
1 Drug
Monoclonal antibody (anti-α4 integrin)
1 Drug
Phosphodiesterase-4 (PDE4) Inhibitor
1 Drug
Sphingosine-1-phosphate (S1P) receptor modulator
1 Drug
TNF-α Inhibitor (Biologic DMARD)
1 Drug
Immunomodulator / Anthelmintic
1 Subclass
Imidazothiazole derivative
1 Drug
Immunomodulatory agent
1 Subclass
Monoclonal antibody – IL-17A antagonist
1 Drug
Immunosuppressant
5 Subclasses
Antimetabolite – Purine analogue
1 Drug
Antimetabolite (Purine synthesis inhibitor)
2 Drugs
Calcineurin Inhibitor
1 Drug
mTOR (mammalian target of rapamycin) inhibitor
1 Drug
Tumour Necrosis Factor (TNF)-α Inhibitor, Chimeric Monoclonal Antibody
1 Drug
Immunosuppressant / Antineoplastic agent
1 Subclass
Mammalian target of rapamycin (mTOR) inhibitor
1 Drug
Immunosuppressant / Biologic Agent
1 Subclass
Tumour Necrosis Factor-alpha (TNF-α) Inhibitor
1 Drug
Immunosuppressant / Cytotoxic agent
1 Subclass
Alkylating agent — Nitrogen mustard derivative
No Drugs
Inotrope
1 Subclass
Phosphodiesterase-3 (PDE3) Inhibitor
1 Drug
Keratolytic Agent
1 Subclass
Topical Antiseborrhoeic / Antipsoriatic
1 Drug
Laxative
5 Subclasses
Osmotic Laxative (Polyether Compound)
1 Drug
Osmotic laxative / Synthetic disaccharide
1 Drug
Stimulant laxative
1 Drug
Stimulant Laxative (Anthraquinone derivative)
1 Drug
Stimulant Laxative (Diphenylmethane derivative)
1 Drug
Laxative / Electrolyte Supplement
1 Subclass
Osmotic Laxative (Saline laxative)
1 Drug
Leukotriene Receptor Antagonist
1 Subclass
Selective Cysteinyl Leukotriene Type-1 (CysLT1) Receptor Blocker
2 Drugs
Lipid-lowering Agent
2 Subclasses
Cholesterol Absorption Inhibitor
1 Drug
HMG-CoA Reductase Inhibitor (Statin)
3 Drugs
Local anaesthetic
1 Subclass
Amide-type local anaesthetic
1 Drug
Mineral Supplement / Antacid
1 Subclass
Calcium salts
1 Drug
Monoclonal Antibody
3 Subclasses
Anti-IgE Monoclonal Antibody
1 Drug
Anti-IL-5 Receptor alpha (anti-IL-5Rα) monoclonal antibody
1 Drug
IL-4 Receptor Alpha Antagonist (Th2 Cytokine Inhibitor)
1 Drug
Mood Stabiliser
1 Subclass
Antimanic Agent
1 Drug
Nasal Decongestant
1 Subclass
Sympathomimetic Alpha-Adrenergic Agonist
1 Drug
Neuromuscular Blockade Reversal Agent
1 Subclass
Selective Relaxant Binding Agent (SRBA)
1 Drug
Neuromuscular Blocking Agent
2 Subclasses
Depolarising Neuromuscular Blocker
1 Drug
Non-depolarising aminosteroid neuromuscular blocker
1 Drug
Non-steroidal Anti-inflammatory Drug (NSAID)
4 Subclasses
Arylacetic acid derivative
1 Drug
Phenylacetic acid derivative
1 Drug
Preferential COX-2 inhibitor (Oxicam derivative)
1 Drug
Selective COX-2 inhibitor
1 Drug
Nonsteroidal Anti-inflammatory Drug (NSAID)
2 Subclasses
Arylacetic acid derivative (Pyrrolizine carboxylic acid derivative)
1 Drug
Propionic Acid Derivative
2 Drugs
Nootropic Agent
1 Subclass
GABA Derivative / Cognition Enhancer
1 Drug
Nutritional Supplement
1 Subclass
Combination Vitamins (with or without Minerals)
1 Drug
Ophthalmic Lubricant
1 Subclass
Ocular Surface Moisturiser
1 Drug
Opioid Analgesic
4 Subclasses
Natural Opiate Alkaloid
1 Drug
Phenanthrene Derivative (Natural Opiate Alkaloid)
1 Drug
Semi-synthetic Opioid (Codeine Derivative)
1 Drug
Synthetic phenylpiperidine opioid
1 Drug
Opioid Antagonist
2 Subclasses
Alcohol and Opioid Dependence Treatment Agent
1 Drug
Pure opioid antagonist
1 Drug
Oral Antidiabetic
1 Subclass
Meglitinide analogue (Glinide)
1 Drug
Osmotic Diuretic
1 Subclass
Hexahydroxy alcohol
1 Drug
Ovulation Inducing Agent
1 Subclass
Selective Estrogen Receptor Modulator (SERM)
2 Drugs
Peripheral Opioid Receptor Antagonist
1 Subclass
Peripherally Acting μ-Opioid Receptor Antagonist (PAMORA)
1 Drug
Phosphate Binder
2 Subclasses
Calcium-based Phosphate Binder
1 Drug
Non-calcium, Non-metal-based Phosphate Binder
1 Drug
Potassium Binder
1 Subclass
Non-polymer Inorganic Cation-exchange Compound
1 Drug
Potassium-binding agent
2 Subclasses
Non-absorbed polymer-based potassium binder
1 Drug
Non-polymer inorganic cation exchanger
1 Drug
Probiotic
1 Subclass
Yeast-based Probiotic
1 Drug
Probiotic Agent
1 Subclass
Gastrointestinal Microflora Modifiers
1 Drug
Prokinetic agent
2 Subclasses
Benzamide derivative (5-HT4 receptor agonist)
1 Drug
Dopamine D2 receptor antagonist (peripheral)
1 Drug
Prokinetic agent / Atypical antipsychotic
1 Subclass
Benzamide derivative (Selective D2 receptor antagonist)
1 Drug
Prokinetic and Antiemetic
1 Subclass
Dopamine D2 Receptor Antagonist
2 Drugs
Prokinetic and Gastrointestinal Motility Agent
1 Subclass
5-HT4 Receptor Partial Agonist
1 Drug
Prostaglandin analogue
2 Subclasses
Prostaglandin E2
1 Drug
Synthetic PGE1 Analogue
1 Drug
Proton Pump Inhibitor (PPI)
3 Subclasses
Benzimidazole Derivative
4 Drugs
Substituted Benzimidazole
3 Drugs
Substituted benzimidazole derivative
1 Drug
Psoralen Photosensitiser
1 Subclass
Skin Disorder Therapy / Melanogenesis Stimulant
1 Drug
Pulmonary vasodilator
1 Subclass
Inhaled selective pulmonary vasodilator gas
1 Drug
Respiratory Agent
1 Subclass
Exogenous Surfactant
1 Drug
Respiratory Agents
1 Subclass
Inhaled Long-Acting β2-Agonist (LABA) + Inhaled Corticosteroid (ICS)
1 Drug
Respiratory Drugs
1 Subclass
Leukotriene Receptor Antagonist + Long-Acting β2-Agonist (LABA)
1 Drug
Respiratory Drugs (Combination Bronchodilator + Anti-inflammatory)
1 Subclass
Long-acting β2-agonist (LABA) + Inhaled Corticosteroid (ICS)
1 Drug
Retinoid
2 Subclasses
Second-generation systemic retinoid
1 Drug
Systemic Retinoid (Vitamin A Derivative)
1 Drug
Retinoid (oral)
1 Subclass
9-cis-Retinoic Acid Derivative
1 Drug
Skeletal Muscle Relaxant
3 Subclasses
Central alpha-2 adrenergic agonist
1 Drug
GABA-A receptor agonist–derived selective muscle relaxant
1 Drug
GABA-B Receptor Agonist
1 Drug
Somatostatin analogue
3 Subclasses
Growth hormone inhibitor / Vasoactive peptide inhibitor
1 Drug
Multireceptor-targeted Somatostatin Analogue
1 Drug
Multireceptor-targeted Somatostatin Analogue / Pituitary Hormone Modulator
No Drugs
Sympathomimetic
1 Subclass
Alpha- and Beta-adrenergic Receptor Agonist
1 Drug
Sympathomimetic agent
1 Subclass
Inotropic vasopressor
1 Drug
Sympathomimetic inotrope
1 Subclass
β1-adrenergic agonist
1 Drug
Thrombolytics
0 Drugs
Thyroid Hormone
1 Subclass
T4 (Thyroxine) Replacement
1 Drug
Urolithiasis Management
1 Subclass
Urinary Alkaliniser / Potassium Salt
1 Drug
Urological Agent
3 Subclasses
Beta-3 Adrenergic Receptor Agonist
1 Drug
Selective α1A-Adrenoceptor Antagonist
1 Drug
β3-Adrenoceptor Agonist
1 Drug
Urological Antispasmodics
1 Subclass
Antimuscarinic (M3-selective)
1 Drug
Uroselective α1-adrenergic receptor antagonist
1 Subclass
α1-blocker (uroselective)
1 Drug
Uterotonic
3 Subclasses
Ergot alkaloid derivative
1 Drug
Long-acting oxytocin analogue
1 Drug
Prostaglandin F2α analogue
2 Drugs
Uterotonic agent
1 Subclass
Ergot alkaloid
1 Drug
Uterotonic hormone
1 Subclass
Posterior pituitary hormone analogue
1 Drug
Vasoconstrictor agent
0 Drugs
Vasodilator
2 Subclasses
Peripheral vasodilator (5-HT2 receptor antagonist)
1 Drug
Prostacyclin (PGI2) Analogue
1 Drug
Vasodilator (Antihypertensive)
1 Subclass
Direct-acting Nitrovasodilator
1 Drug
Vasodilator and Antiplatelet Agent
1 Subclass
Phosphodiesterase III Inhibitor
1 Drug
Vasodilators for Pulmonary Hypertension
1 Subclass
Prostacyclin Analogue
1 Drug
Vasopressin Analogue
1 Drug
Antidiuretic Hormone (ADH) Analogue
1 Drug
Terlipressin
Vasopressin receptor antagonist
1 Subclass
Non-selective V1A and V2 receptor antagonist
1 Drug
Vasopressin Receptor Antagonist (Vaptan)
1 Subclass
Selective V2-Receptor Antagonist
1 Drug
Vasopressor / Antidiuretic Hormone
1 Subclass
Arginine Vasopressin Analog
1 Drug
Vitamin
2 Subclasses
Water-soluble vitamin (Vitamin B1)
1 Drug
Water-soluble vitamin (Vitamin C)
1 Drug
Vitamin / Nutritional supplement
1 Subclass
Fat-soluble vitamin
1 Drug
Vitamin D analog
2 Subclasses
Active vitamin D3 (1,25-dihydroxycholecalciferol)
1 Drug
Topical antipsoriatic agent
1 Drug
Vitamin D analogue
1 Subclass
Active vitamin D (1α-hydroxylated form)
1 Drug
Vitamin supplement
1 Subclass
Water-soluble vitamin (Vitamin B6)
1 Drug
Xanthine oxidase inhibitor
1 Drug
Uric acid lowering agent
1 Drug
Febuxostat